2. Signaling Pathways
  3. Vitamin D Related/Nuclear Receptor
  4. Estrogen Receptor/ERR
  5. Estrogen Receptor/ERR Chemical

Estrogen Receptor/ERR Chemical

Estrogen Receptor/ERR Isoform Comparison

Estrogen Receptor/ERR Chemicals (2):

Cat. No. Product Name Effect Purity
  • HY-117726
    WAY-169916
    		Chemical 99.60%
    WAY-169916 is a pathway-selective ligand of ER (estrogen receptor) that acts by inhibiting NF-kB transcriptional activity. WAY-169916 has potent anti-inflammatory effect.
  • HY-103453
    (R)-DPN
    		Chemical
    (R)-DPN (compound 3) is a selective ERβ ligand with EC50s of 2.9, 0.8 nM for ERα and ERβ, respectively. (R)-DPN shows a very high affinity and potency preference for ERβ over ERα. (R)-DPN shows cytoxicity for HEC-1 and U2OS cells with EC50s of 286, 205 nM, respectively.